Cymbopogon citratus, or lemongrass, is renowned for its aromatic properties and its extensive use in traditional medicine, cosmetics, and culinary preparations. A rich source of essential electrolytes, minerals, vitamins, macronutrients, and phytochemicals, lemongrass offers a wide range of biological and therapeutic advantages. These effects are mediated by bioactive compounds, including geranial, nerol, and myrcene, which have been demonstrated to exert anti-inflammatory, antifungal, antineoplastic, and antibacterial properties. Additionally, the high phenolic content in lemongrass contributes to its antioxidant capacity, neutralizing free radicals, chelating metal ions, and inhibiting radical-producing enzymes. Lemongrass has also demonstrated hepatoprotective effects and the capacity to enhance cardiovascular health. The extracts have been observed to possess analgesic properties, which are primarily attributable to the presence of citral. This provides pain relief by inhibiting inflammation and interacting with opioid receptors, thereby offering natural alternatives for pain management. Furthermore, lemongrass facilitates digestion by stimulating enzyme production, alleviating gastrointestinal discomfort, and preventing gastric ulcers through mucin production and reduced acid secretion. While lemongrass has garnered scientific interest due to its efficacy, health benefits, and minimal side effects, caution is warranted in the use of lemongrass extracts, infusions, and essential oils, particularly in direct skin application and in combination with certain medications due to potential interactions. Proper dosage and moderation are essential to avoid adverse effects. Further research is required to determine the characteristics and potential adverse effects associated with the use of lemongrass. The combination of traditional practices with modern evidence-based scientific knowledge serves to highlight the potential of lemongrass in the development of sustainable and holistic health solutions.